Small Molecule Potentiator to Enhance the Efficacy of Cancer Immunotherapy

BACKGROUND

Cancer immune surveillance depends on dynamic stepwise interactions between immunogenic tumors and cells of the innate and adaptive immune system. Researchers at the University of Calgary investigated the microbiome-mediated modulation of the host tumor immune surveillance using mouse models, and discovered a class of microbiome-derived metabolites that modulate gene expression of the immune cells within tumor microenvironment, ultimately increase tumor-specific CD8+ T cells within tumor microenvironment and enhance tumor immune surveillance in mice and synergizes with immune checkpoint blockade therapy.

AREAS OF APPLICATION

Cancer Immune therapy

  • Potential compounds for improved checkpoint blockade therapy efficacy
  • Potential to serve as molecular marker for cancer immune therapy
  • Potential as new nutraceutical

COMPETITIVE ADVANTAGES

  • Natrual product – safety level is high
  • The metabolites synergistically with clinically approved immune checkpoint blockades to improve overall survival rates (from 0 survival after 20 days to over 25% survival after 60 days).
  • The metabolites work independent of the host microbiome composition when used as systemic treatment.
  • Potential target and immune functional pathway identified, mouse model and cell lines established

STAGE OF DEVELOPMENT

In vitro and in vivo preclinical data.

INTELLECTUAL PROPERTY STATUS

PCT application filed.